8 results for "other-nuclear-receptor-inhibitors&view=expanded" in Products

COUP-TFII inhibitor

Chemical Name: N-[2-(3,4-Dimethoxyphenyl)ethyl]-6-methylthieno[2,3-d]pyrimidin-4-amine hydrochloride
Purity: ≥98%
COUP-TFII inhibitor
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Steroid receptor coactivator 3 (SRC-3) inhibitor

Chemical Name: 1-(2-Pyridinyl)ethanone 2-(1-methyl-1H-benzimidazol-2-yl)hydrazone hydrochloride
Purity: ≥98%
Steroid receptor coactivator 3 (SRC-3) inhibitor
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Nuclear receptor-binding SET domain (NSD) 3 antagonist; selectively binds PWWP1 domain

Chemical Name: (4-(5-(7-Fluoroquinolin-4-yl)-1-methyl-1H-imidazol-4-yl)-3,5-dimethylphenyl)methanamine trihydrochloride
Purity: ≥98%
Nuclear receptor-binding SET domain (NSD) 3 antagonist; selectively binds PWWP1 domain
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NSD2 Degrader (PROTAC®)

Chemical Name: N-Cyclopropyl-N-(4-((5-(3-(2-((2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindolin-4-yl)amino)acetamido)propoxy)pyridin-2-yl)-carbamoyl)benzyl)-3-oxo-3,4-dihydro-2H-benzo[b][1,4]oxazine-7-carboxamide
Purity: ≥98%
NSD2 Degrader (PROTAC®)
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Nur77 antagonist

Chemical Name: 1,1-Bis(3'-indolyl)-1-(p-hydroxyphenyl)methane
Purity: ≥98%
Nur77 antagonist
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Nurr1 activator; inhibits NF-κB-dependent gene expression

Chemical Name: 3,3'-[(4-Chlorophenyl)methylene]bis[1H-indole]
Purity: ≥98%
Nurr1 activator; inhibits NF-κB-dependent gene expression
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Selective steroidogenic factor-1 (SF-1, NR5A1) inhibitor

Chemical Name: Ethyl 2-[[2-[2-[(2,3-Dihydro-1,4-benzodioxin-6-yl)amino]-2-oxoethyl]-1,2-dihydro-1-oxo-5-isoquinolinyl]oxy]propanoate
Purity: ≥98%
Selective steroidogenic factor-1 (SF-1, NR5A1) inhibitor
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Progesterone receptor membrane component 1 (Pgrmc1) ligand

Chemical Name: cis-2-[[1-(4-Chlorophenyl)-1H-tetrazol-5-yl]thio]-1-(1,2,3,4,4a,9b-hexahydro-2,8-dimethyl-5H-pyrido[4,3-b]indol-5-yl)-ethanone
Purity: ≥97%
Progesterone receptor membrane component 1 (Pgrmc1) ligand
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