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Potent and selective cereblon Degrader (PROTAC®); cell-permeable
(+)-JQ1 based Degrader (PROTAC®) that selectively degrades BRD4
(+)-JQ1 based Degrader (PROTAC®) targeting BET bromodomains, active in vivo
Homo-PROTAC® for self-degradation of pVHL30
Potent and selective BRD9 Degrader (PROTAC®)
Potent BRD9 Degrader (PROTAC®)
Potent and selective androgen receptor PROTAC®
Selective peptide-based β-catenin Degrader (PROTAC®)
(+)-JQ1 based PROTAC® with selectivity for BRD4
Multikinase Degrader (PROTAC®)
Selective Cdk4/6 Degrader (PROTAC®)
Potent and selective (+)-JQ1 based Degrader (PROTAC®) targeting BET bromodomains, active in vivo
Potent and selective BTK Degrader (PROTAC®)
Potent and selective Wee1 Degrader (PROTAC®)
Potent BET bromodomain PROTAC®; also degrades BRD-tagged chimeric antigen receptors (CAR) in T cells
Potent TANK-binding kinase 1 (TBK1) PROTAC®
Potent EGFR PROTAC®; also degrades HER2
c-MET PROTAC®; also degrades exon-14-deleted c-MET
Potent and selective p38α PROTAC®
Potent and selective VHL-recruiting Degrader (PROTAC®) of mutant EGFR
Selective BRAF-V600E protein Degrader (uSMITE™)
Potent and selective EP300 Degrader
TRIM24 Degrader (PROTAC®)
Potent and selective BRD4 Degrader (PROTAC®)
Selective ALK Degrader (PROTAC®)
Selective ALK Degrader (PROTAC®)
Selective Cdk6 Degrader (PROTAC®)
Potent and selective BRD7/9 Degrader (PROTAC®)
Selective Cdk4 Degrader (PROTAC®)
Potent and selective ERα Degrader (SNIPER)
Potent and selective p38α and p38β Degrader (PROTAC®); active in vivo
Cereblon Degrader (PROTAC®)
Potent and selective p38δ PROTAC®
Selective α1A adrenergic receptor Degrader (PROTAC®)
Photoswitchable BET bromodomain Degrader (PHOTAC)
SRC-1 peptide-based PROTAC®; active in vivo
Selective and potent TAG Degrader for auxin-inducible degron 2 system
Potent and selective cereblon-recruiting Degrader (PROTAC®) of mutant EGFR
Potent tropomyosin receptor kinase (TRK) degrader
Potent and selective trivalent BET Bromodomain Degrader (PROTAC®)
Negative control for SJF 0628 (Cat. No. 7463)
Potent MIF Degrader (PROTAC®)
Selective CDK12 PROTAC® Degrader
Degrades mutant FKBP12F36V fusion proteins; useful alternative to genetic methods for target validation