10 results for "Adenosine A2aR" in Products
Adenosine A2aR Products
Adenosine A2A Receptor (ADORA2A, Adenosine A2aR) is one of several receptor subtypes for adenosine. The activity of Adenosine A2aR, a G protein-coupled receptor family member, is mediated by G proteins which activate adenylyl cyclase. Adenosine A2aR is abundant in basal ganglia, vasculature and platelets and is a major target of caffeine. Variability in the acute blood pressure response to coffee may be partly explained by genetic polymorphisms of the adenosine A2A receptors, including Adenosine A2aR, and alpha(2)-adrenergic receptors.
Potent and highly selective A2A antagonist
| Chemical Name: | 4-(2-[7-Amino-2-(2-furyl)[1,2,4]triazolo[2,3-a][1,3,5]triazin-5-ylamino]ethyl)phenol |
| Purity: | ≥98% |
Potent, highly selective A2A antagonist
| Chemical Name: | 2-(2-Furanyl)-7-(2-phenylethyl)-7H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-amine |
| Purity: | ≥98% |
Very selective, high affinity A2A antagonist
| Chemical Name: | 2-(2-Furanyl)-7-[3-(4-methoxyphenyl)propyl]-7H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-amine |
| Purity: | ≥98% |
A1 and A2B antagonist. CNS stimulant
| Chemical Name: | 3,7-Dihydro-1,3,7-trimethyl-1H-purine-2,6-dione |
| Purity: | ≥98% |
Potent adenosine receptor antagonist
| Chemical Name: | 9-Chloro-2-(2-furanyl)-[1,2,4]triazolo[1,5-c]quinazolin-5-amine |
| Purity: | ≥98% |
Potent and selective A2A antagonist
| Alternate Names: | KW-6002 |
| Chemical Name: | 8-[(1E)-2-(2-(3,4-Dimethoxyphenyl)ethenyl]-1,3-diethyl-3,7-dihydro-7-methyl-1H-purine-2,6-dione |
| Purity: | ≥98% |
Adenosine A2A antagonist
| Chemical Name: | 8-Ethoxy-9-ethyl-9H-purin-6-amine |
| Purity: | ≥98% |
Adenosine receptor antagonist
| Chemical Name: | 2-[4-(2,3,6,7-Tetrahydro-2,6-dioxo-1,3-dipropyl-1H-purin-8-yl)phenoxy]-acetic acid |
| Purity: | ≥98% |
Adenosine receptor antagonist
| Alternate Names: | Xanthine amine congener |
| Chemical Name: | N-(2-Aminoethyl)-2-[4-(2,3,6,7-tetrahydro-2,6-dioxo-1,3-dipropyl-1H-purin-8-yl)phenoxy]-acetamide dihydrochloride |
| Purity: | ≥98% |
Potent and selective A2A antagonist
| Chemical Name: | N-[2-(3,5-Dimethyl-1H-pyrazol-1-yl)-6-[6-(4-methoxy-1-piperidinyl)-2-pyridinyl]-4-pyrimidinyl]acetamide |
| Purity: | ≥98% |
