12 results for "rho-gtpase-inhibitors&view=expanded" in Products

Selective inhibitor of Rac1-GEF interaction; antioncogenic

Chemical Name: N6-[2-[[4-(Diethylamino)-1-methylbutyl]amino]-6-methyl-4-pyrimidinyl]-2-methyl-4,6-quinolinediamine trihydrochloride
Purity: ≥98%
Selective inhibitor of Rac1-GEF interaction; antioncogenic
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Potent Rac family inhibitor

Chemical Name: 5-(5-(7-(Trifluoromethyl)quinolin-4-ylthio)pentyloxy)-2-(morpholinomethyl)-4H-pyran-4-one dihydrochloride
Purity: ≥98%
Potent Rac family inhibitor
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Selective Cdc42 Rho family inhibitor

Alternate Names: CID 2950007
Chemical Name: 4-[4,5-Dihydro-5-(4-methoxyphenyl)-3-phenyl-1H-pyrazol-1-yl]benzenesulfonamide
Purity: ≥98%
Selective Cdc42 Rho family inhibitor
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Rho inhibitor

Chemical Name: D-Tryptophan (2E)-2-(6-quinoxalinylmethylene)hydrazide hydrochloride
Purity: ≥98%
Rho inhibitor
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DOCK2-Rac1 interaction inhibitor

Chemical Name: 4-[3-(2-Chlorophenyl)-2-propen-1-ylidene]-1-phenyl-3,5-pyrazolidinedione
Purity: ≥98%
DOCK2-Rac1 interaction inhibitor
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Cdc42 inhibitor

Chemical Name: 2-[(2,3,4,9-Tetrahydro-6-phenyl-1H-carbazol-1-yl)amino]ethanol
Purity: ≥98%
Cdc42 inhibitor
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Promotes mitochondrial Rho GTPase 1 (Miro1) degradation

Chemical Name: N-(3-Fluorophenyl)-N'-[4-[[6-(1H-imidazol-1-yl)-4-pyrimidinyl]amino]phenyl]urea hydrochloride
Purity: ≥98%
Promotes mitochondrial Rho GTPase 1 (Miro1) degradation
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Rac inhibitor

Chemical Name: N4-(9-Ethyl-9H-carbazol-3-yl)-N2-[3-(4-morpholinyl)propyl]-2,4-pyrimidinediamine
Purity: ≥98%
Rac inhibitor
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Potent and selective CSN5 (COP9 signalosome) inhibitor

Chemical Name: 3-(Difluoromethyl)-N-(6-((5S,6S)-6-hydroxy-6,7,8,9-tetrahydro-5H-imidazo[1,5-a]azepin-5-yl)-[1,10-biphenyl]-3-yl)-1-isopropyl-1H-pyrazole-5-carboxamide
Purity: ≥98%
Novartis vs Bio-Techne batch comparison for CSN5i-3
(2)
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Rac1 inhibitor; blocks Rac1-P-Rex1 interaction

Chemical Name: N-(3,5-Dimethylphenyl)-N'-[2-(trifluoromethyl)phenyl]guanidine
Purity: ≥98%
Rac1 inhibitor; blocks Rac1-P-Rex1 interaction
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