Histamine H1 Receptor Antagonists: Products

Histamine H1R (HRH1) is a G-protein coupled 7-transmembrane putative glycoprotein that is implicated in the pathogenesis of asthma and is a major pharmaceutical target for antihistamines.

"Histamine H1 Receptor Antagonists" has 17 results in Products.
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(S)-(+)-Dimethindene maleate 

M2-selective antagonist

Clemastine fumarate 

H1 antagonist

Ketotifen fumarate 

H1 antagonist

Mirtazapine 

Potent 5-HT2 antagonist; also 5-HT3, H1 and α2 antagonist; antidepressant

Astemizole 

Orally active, potent H1 antagonist. Also KV11.1 (hERG) channel blocker

Cetirizine dihydrochloride 

Selective H1 antagonist

Terfenadine 

H1 antagonist. Also KV11.1 (hERG) and Kir6 (KATP) channel blocker

Doxepin hydrochloride 

Highly potent H1 antagonist. Also binds to H4 receptor

trans-Triprolidine hydrochloride 

Standard H1 antagonist, highly potent

Loratidine 

Peripheral H1 antagonist; antiallergic agent

Fexofenadine hydrochloride 

H1 receptor antagonist; non-sedating antiallergic agent

Diphenhydramine hydrochloride 

H1 receptor antagonist

Zotepine 

5-HT2A/D2 antagonist; atypical antipsychotic

Olopatadine hydrochloride 

H1 antagonist; ocular antiallergic agent

Meclizine dihydrochloride 

Human pregnane X receptor agonist; H1 antagonist

Clemizole hydrochloride 

TRPC5 blocker; also H1 antagonist

Desloratadine 

High affinity H1 antagonist; anti-inflammatory
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