Histamine H1 Receptor Antagonists: Products

Histamine H1R (HRH1) is a G-protein coupled 7-transmembrane putative glycoprotein that is implicated in the pathogenesis of asthma and is a major pharmaceutical target for antihistamines.

"Histamine H1 Receptor Antagonists" has 17 results in Products.
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(S)-(+)-Dimethindene maleate

M2-selective antagonist

Clemastine fumarate

H1 antagonist

Mirtazapine

Potent 5-HT2 antagonist; also 5-HT3, H1 and α2 antagonist; antidepressant

Ketotifen fumarate

H1 antagonist

Astemizole

Orally active, potent H1 antagonist. Also KV11.1 (hERG) channel blocker

Terfenadine

H1 antagonist. Also KV11.1 (hERG) and Kir6 (KATP) channel blocker

Meclizine dihydrochloride

Human pregnane X receptor agonist; H1 antagonist

Doxepin hydrochloride

Highly potent H1 antagonist. Also binds to H4 receptor

trans-Triprolidine hydrochloride

Standard H1 antagonist, highly potent

Loratidine

Peripheral H1 antagonist; antiallergic agent

Fexofenadine hydrochloride

H1 receptor antagonist; non-sedating antiallergic agent

Cetirizine dihydrochloride

Selective H1 antagonist

Diphenhydramine hydrochloride

H1 receptor antagonist

Zotepine

5-HT2A/D2 antagonist; atypical antipsychotic

Olopatadine hydrochloride

H1 antagonist; ocular antiallergic agent

Clemizole hydrochloride

TRPC5 blocker; also H1 antagonist

Desloratadine

High affinity H1 antagonist; anti-inflammatory
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