13 results for "PI 3-Kinase Inhibitors" in Products

PI 3-Kinase Inhibitors

Inhibitor of PI 3-kinase, mTOR and DNA-PK

Chemical Name: 3-[4-(4-Morpholinylpyrido[3',2':4,5]furo[3,2-d]pyrimidin-2-yl]phenol hydrochloride
Purity: ≥98%
Inhibitor of PI 3-kinase, mTOR and DNA-PK
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PI 3-kinase inhibitor, more potent than LY 294002 (Cat. No. 1130)

Chemical Name: 2-(4-Morpholinyl)-8-(4-aminopheny)l-4H-1-benzopyran-4-one
Purity: ≥98%
PI 3-kinase inhibitor, more potent than LY 294002 (Cat. No. 1130)
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Prototypical PI 3-kinase inhibitor; also inhibits other kinases

Chemical Name: 2-(4-Morpholinyl)-8-phenyl-4H-1-benzopyran-4-one hydrochloride
Purity: ≥99%
Prototypical PI 3-kinase inhibitor; also inhibits other kinases
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Potent, irreversible inhibitor of PI 3-kinase. Also inhibitor of PLK1

Alternate Names: SL-2052
Chemical Name: (1S,6bR,9aS,11R,11bR) 11-(Acetyloxy)-1,6b,7,8,9a,10,11,11b-octahydro-1-(methoxymethyl)-9a,11b-dimethyl-3H-furo[4,3,2-de]indeno[4,5,-h]-2-h]-2-benzopyran-3,6,9-trione
Purity: ≥98%
Potent, irreversible inhibitor of PI 3-kinase. Also inhibitor of PLK1
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Non-selective PI 3-kinase inhibitor

Chemical Name: 2-(3,4-Dihydroxyphenyl)-3,5,7-trihydroxy-4H-1-benzopyran-4-one
Purity: ≥98%
Non-selective PI 3-kinase inhibitor
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Potent and selective PI 3-Kβ inhibitor

Chemical Name: (-)-2-[[(1R)-1-[7-Methyl-2-(4-morpholinyl)-4-oxo-4H-pyrido[1,2-a]pyrimidin-9-yl]ethyl]amino]benzoic acid
Purity: ≥98%
Potent and selective PI 3-Kβ inhibitor
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PI 3-K/Akt/mTOR signaling inhibitor; blocks phosphorylation of Akt and p70S6K in vitro

Chemical Name: 3,8-Dihydroxy-6H-dibenzo[b,d]pyran-6-one
Purity: ≥98%
PI 3-K/Akt/mTOR signaling inhibitor; blocks phosphorylation of Akt and p70S6K in vitro
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Potent and selective PI 3-kinase p110α inhibitor

Chemical Name: (2S)-N1-[2-(1,1-Dimethylethyl)-4'-methyl[4,5'-bithiazol]-2'-yl]-1,2-pyrrolidinedicarboxamide
Purity: ≥98%
Potent and selective PI 3-kinase p110α inhibitor
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Highly potent PI 3-kinase inhibitor; also potent inhibitor of mTOR and DNA-PK

Alternate Names: GSK2126458
Chemical Name: 2,4-Difluoro-N-[2-methoxy-5-[4-(4-pyridazinyl)-6-quinolinyl]-3-pyridinyl]benzenesulfonamide
Purity: ≥98%
Highly potent PI 3-kinase inhibitor; also potent inhibitor of mTOR and DNA-PK
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Class III PI 3-kinase inhibitor; also inhibits autophagy

Alternate Names: 3-MA
Chemical Name: 3-Methyl-3H-purin-6-amine
Purity: ≥98%
Class III PI 3-kinase inhibitor; also inhibits autophagy
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Potent PI 3-Kinase δ isoform inhibitor

Chemical Name: 5-Fluoro-3-phenyl-2-[(1S)-1-(9H-purin-6-ylamino)propyl]-4(3H)-quinazolinone
Purity: ≥98%
Potent PI 3-Kinase δ isoform inhibitor
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Potent PI3K inhibitor, also used in hPSCs mesendoderm differentiation

Chemical Name: N-(2,3-Dihydro-7,8-dimethoxyimidazo[1,2-c]quinazolin-5-yl)-3-pyridinecarboxamide
Purity: ≥98%
Potent PI3K inhibitor, also used in hPSCs mesendoderm differentiation
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Potent pan-class I PI3 kinase inhibitor

Chemical Name: 2-(1H-Indazol-4-yl)-6-[[4-(methylsulfonyl)-1-piperazinyl]methyl]-4-(4-morpholinyl)-thieno[3,2-d]pyrimidine
Purity: ≥98%
Potent pan-class I PI3 kinase inhibitor
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