16 results for "VEGF-Receptor-Inhibitors" in Products

VEGFR inhibitor. Also inhibits KIT, RET, MET and FLT3

Alternate Names: Semaxinib
Chemical Name: 3-[(3,5-Dimethyl-1H-pyrrol-2-yl)methylene]-1,3-dihydro-2H-indol-2-one
Purity: ≥98%
VEGFR inhibitor. Also inhibits KIT, RET, MET and FLT3
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Potent FGFR and VEGFR inhibitor

Alternate Names: PF-02969207,PNU-0290908
Chemical Name: 2-[(1,2-Dihydro-2-oxo-3H-indol-3-ylidene)methyl]-4-methyl-1H-pyrrole-3-propanoic acid
Purity: ≥95%
Potent FGFR and VEGFR inhibitor
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Potent, selective inhibitor of VEGFR-2

Chemical Name: 5-((7-Benzyloxyquinazolin-4-yl)amino)-4-fluoro-2-methylphenol hydrochloride
Purity: ≥98%
Potent, selective inhibitor of VEGFR-2
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Potent VEGFR, PDGFR and FGFR inhibitor

Chemical Name: Methyl (Z)-3-[[[4-(N-methyl-2-(4-methylpiperazin-1-yl)acetamido)phenyl)amino)(phenyl)methylene]-2-oxoindoline-6-carboxylate
Purity: ≥98%
Potent VEGFR, PDGFR and FGFR inhibitor
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Potent, selective VEGFR-2 inhibitor

Chemical Name: N-(2,4-Difluorophenyl)-N'-[4-[(6,7-dimethoxy-4-quinolinyl)oxy]-2-fluorophenyl]urea
Purity: ≥97%
Potent, selective VEGFR-2 inhibitor
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Potent VEGFR-1, -2 and -3 inhibitor

Chemical Name: N-Methyl-[[3[(1E)-2-(2-pyridinyl)ethenyl]-1H-indazol-6-yl]thio]-benzamide
Purity: ≥98%
Potent VEGFR-1, -2 and -3 inhibitor
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Potent VEGFR inhibitor; also inhibits other RTKs

Alternate Names: Cabozantinib,BMS 907351
Chemical Name: N-[4-[(6,7-Dimethoxy-4-quinolinyl)oxy]phenyl]-N-(4-fluorophenyl)-1,1-cyclopropanedicarboxamide
Purity: ≥98%
Potent VEGFR inhibitor; also inhibits other RTKs
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Potent VEGFR, PDGFRβ and KIT inhibitor

Alternate Names: SU 11248
Chemical Name: N-[2-(Diethylamino)ethyl]-5-[(Z)-(5-fluoro-1,2-dihydro-2-oxo-3H-indol-3-ylidine)methyl]-2,4-dimethyl-1H-pyrrole-3-carboxamide (2S)-2-hydroxybutanedioate salt
Purity: ≥98%
Potent VEGFR, PDGFRβ and KIT inhibitor
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Potent inhibitor of VEGFR, PDGFR and FGFR

Chemical Name: 4-[(4-Fluoro-2-methyl-1H-indol-5-yl)oxy]-6-methoxy-7-[3-(1-pyrrolidinyl)propoxy]quinazoline
Purity: ≥98%
Potent inhibitor of VEGFR, PDGFR and FGFR
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Potent VEGFR-2 inhibitor, also inhibits EGFR and RET oncoproteins activity

Chemical Name: N-(4-Bromo-2-fluorophenyl)-6-methoxy-7-[(1-methyl-4-piperidinyl)methoxy]-4-quinazolinamine
Purity: ≥98%
Potent VEGFR-2 inhibitor, also inhibits EGFR and RET oncoproteins activity
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