15 results for "VEGF Receptor Inhibitors" in Products

VEGF Receptor Inhibitors

Vascular endothelial growth factor is a signaling protein involved in the regulation of angiogenesis and vasculogenesis.

Whilst multiple receptors and ligands are involved in angiogenesis, VEGF signaling is one of the most important, rate-limiting steps of the process. VEGF is diffusible and selective for vascular endothelial cells, and possesses the ability to promote the growth and survival of these cells in vitro. Hypoxic conditions activate hypoxia-inducible factor 1 (HIF-1), resulting in ...

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Potent FGFR and VEGFR inhibitor

Alternate Names: PF-02969207,PNU-0290908
Chemical Name: 2-[(1,2-Dihydro-2-oxo-3H-indol-3-ylidene)methyl]-4-methyl-1H-pyrrole-3-propanoic acid
Purity: ≥95%
Potent FGFR and VEGFR inhibitor
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VEGFR inhibitor. Also inhibits KIT, RET, MET and FLT3

Alternate Names: Semaxinib
Chemical Name: 3-[(3,5-Dimethyl-1H-pyrrol-2-yl)methylene]-1,3-dihydro-2H-indol-2-one
Purity: ≥98%
VEGFR inhibitor. Also inhibits KIT, RET, MET and FLT3
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Potent, selective inhibitor of VEGFR-2

Chemical Name: 5-((7-Benzyloxyquinazolin-4-yl)amino)-4-fluoro-2-methylphenol hydrochloride
Purity: ≥98%
Potent, selective inhibitor of VEGFR-2
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Potent VEGFR, PDGFR and FGFR inhibitor

Chemical Name: Methyl (Z)-3-[[[4-(N-methyl-2-(4-methylpiperazin-1-yl)acetamido)phenyl)amino)(phenyl)methylene]-2-oxoindoline-6-carboxylate
Purity: ≥98%
Potent VEGFR, PDGFR and FGFR inhibitor
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Potent, selective VEGFR-2 inhibitor

Chemical Name: N-(2,4-Difluorophenyl)-N'-[4-[(6,7-dimethoxy-4-quinolinyl)oxy]-2-fluorophenyl]urea
Purity: ≥97%
Potent, selective VEGFR-2 inhibitor
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Potent Raf-1 inhibitor; also inhibits VEGFR-2, VEGFR-3, PDGFR-β, Flt-3 and cKIT

Chemical Name: 4-[4-[[[[4-Chloro-3-(trifluoromethyl)phenyl]amino]carbonyl]amino]phenoxy]-N-methyl-2-pyridinecarboxamide
Purity: ≥98%
Potent Raf-1 inhibitor; also inhibits VEGFR-2, VEGFR-3, PDGFR-β, Flt-3 and cKIT
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Neuropilin 1 (NRP1) receptor antagonist; inhibits VEGFA binding to NRP1

Chemical Name: N2-[[3-[(2,1,3-Benzothiadiazol-4-ylsulfonyl)amino]-2-thienyl]carbonyl]-L-arginine trifluoroacetate
Purity: ≥98%
Neuropilin 1 (NRP1) receptor antagonist; inhibits VEGFA binding to NRP1
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Potent VEGFR, PDGFRβ and KIT inhibitor

Alternate Names: SU 11248
Chemical Name: N-[2-(Diethylamino)ethyl]-5-[(Z)-(5-fluoro-1,2-dihydro-2-oxo-3H-indol-3-ylidine)methyl]-2,4-dimethyl-1H-pyrrole-3-carboxamide (2S)-2-hydroxybutanedioate salt
Purity: ≥98%
Potent VEGFR, PDGFRβ and KIT inhibitor
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Potent multi-kinase and pan-Bcr-Abl inhibitor

Alternate Names: Ponatinib
Chemical Name: 3-(2-Imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-N-[4-[(4-methyl-1-piperazinyl)methyl]-3-(trifluoromethyl)phenyl]-benzamide
Purity: ≥98%
Potent multi-kinase and pan-Bcr-Abl inhibitor
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Potent VEGFR-1, -2 and -3 inhibitor

Chemical Name: N-Methyl-[[3[(1E)-2-(2-pyridinyl)ethenyl]-1H-indazol-6-yl]thio]-benzamide
Purity: ≥98%
Potent VEGFR-1, -2 and -3 inhibitor
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Potent EGFR and VEGFR inhibitor

Chemical Name: 6-[4-[(4-Ethyl-1-piperazinyl)methyl]phenyl]-N-[(1R)-1-phenylethyl]-7H-pyrrolo[2,3-d]pyrimidin-4-amine
Purity: ≥98%
Potent EGFR and VEGFR inhibitor
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Potent VEGFR inhibitor; also inhibits other RTKs

Alternate Names: Cabozantinib,BMS 907351
Chemical Name: N-[4-[(6,7-Dimethoxy-4-quinolinyl)oxy]phenyl]-N-(4-fluorophenyl)-1,1-cyclopropanedicarboxamide
Purity: ≥98%
Potent VEGFR inhibitor; also inhibits other RTKs
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Potent VEGFR inhibitor; also aromatase inhibitor

Alternate Names: CGP 79787D,PTK787/ZK222584
Chemical Name: N-(4-Chlorophenyl)-4-(4-pyridinylmethyl)-1-phthalazinamine succinate
Purity: ≥98%
Potent VEGFR inhibitor; also aromatase inhibitor
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Potent inhibitor of VEGFR, PDGFR and FGFR

Chemical Name: 4-[(4-Fluoro-2-methyl-1H-indol-5-yl)oxy]-6-methoxy-7-[3-(1-pyrrolidinyl)propoxy]quinazoline
Purity: ≥98%
Potent inhibitor of VEGFR, PDGFR and FGFR
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Potent VEGFR-2 inhibitor, also inhibits EGFR and RET oncoproteins activity

Chemical Name: N-(4-Bromo-2-fluorophenyl)-6-methoxy-7-[(1-methyl-4-piperidinyl)methoxy]-4-quinazolinamine
Purity: ≥98%
Potent VEGFR-2 inhibitor, also inhibits EGFR and RET oncoproteins activity
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