200 results for "PARP" in Products

PARP Products

PARP [Poly(ADP-ribose) Polymerase], also known as ADPRT and PPOL, is a 118-kDa enzyme that uses NAD as a substrate to catalyze the covalent transfer of ADP-ribose to a variety of nuclear protein acceptors. ADP ribosyltransferase is required for cellular repair, and PARP expression is induced by single-strand breaks in DNA. PARP is proteolytically cleaved by Caspase-3 into two fragments of 89- and 24-kDa in one of the hallmark events of apoptosis.

Potent tankyrase inhibitor

GMP Version Available: TB3748-GMP
GMP
Alternate Names: XAV939 Wnt Signaling Inhibitor
Chemical Name: 3,5,7,8-Tetrahydro-2-[4-(trifluoromethyl)phenyl]-4H-thiopyrano[4,3-d]pyrimidin-4-one
Purity: ≥98%
Potent tankyrase inhibitor
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Reactivity: Human, Mouse, Rat (Negative)
Details: Mouse IgG2b Kappa Monoclonal Clone #194C1439
Applications: WB, Flow, ICC/IF, CyTOF-ready
Western Blot: PARP Antibody (194C1439)CleavedAzide and BSA Free [NBP2-27335]
(3)
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Reactivity: Human, Mouse, Rat (Negative)
Details: Mouse IgG2b Kappa Monoclonal Clone #194C1439
Applications: WB, Flow, ICC/IF
Western Blot: PARP Antibody (194C1439)CleavedBSA Free [NB100-56599]
(3)
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Reactivity: Human, Mouse
Details: Rabbit IgG Polyclonal
Applications: IHC, WB, ICC/IF, Mycoplasma
Western Blot: PARP Antibody [NBP2-13732]
(7)
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Reactivity: Human
Details: Mouse IgG1 Monoclonal Clone #CL2220
Applications: IHC, WB, ICC/IF, Mycoplasma
Western Blot: PARP Antibody (CL2220) [NBP2-36747]
(10)
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XAV 939 synthesized to cGMP guidelines

Chemical Name: 3,5,7,8-Tetrahydro-2-[4-(trifluoromethyl)phenyl]-4H-thiopyrano[4,3-d]pyrimidin-4-one
Purity: ≥99%
XAV 939 synthesized to cGMP guidelines
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Recombinant Monoclonal Antibody

Reactivity: Human, Mouse, Rat
Details: Rabbit IgG Monoclonal Clone #2G8N7
Applications: IHC, ELISA, ICC/IF
PARP Antibody (2G8N7)
(14)
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Reactivity: Human
Details: Mouse IgG1 Monoclonal Clone #CL2209
Applications: IHC, WB, Mycoplasma
Western Blot: PARP Antibody (CL2209) [NBP2-36748]
(7)
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Reactivity: Human
Details: Mouse IgG1 Monoclonal Clone #CL2220
Applications: IHC, WB, ICC/IF
PARP Antibody (CL2220) - Azide and BSA Free Immunocytochemistry/ Immunofluorescence: PARP Antibody [NBP3-44461]
(10)
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Biotinylated-NAD+; substrate for ADP-ribosylation

Chemical Name: β-Nicotinamide-N6-[2-[[6-[biotinyl]amino]hexyl]amino]-2-oxoethyl]adenine dinucleotide
Biotinylated-NAD+; substrate for ADP-ribosylation
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PARP-1 inhibitor

Chemical Name: Pyridine-3-carboxamide
Purity: ≥99%
iPSC-derived Human Intestinal Organoid
(5)
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Reactivity: Human
Details: Mouse IgG1 Monoclonal Clone #CL2209
Applications: IHC, WB
PARP Antibody (CL2209) - Azide and BSA Free Immunohistochemistry-Paraffin: PARP Antibody [NBP3-44462]
(7)
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Recombinant Monoclonal Antibody

Reactivity: Human
Details: Rabbit IgG Monoclonal Clone #8C7
Applications: IHC, WB, ELISA, Flow, ICC/IF
PARP Antibody (8C7)
(5)
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Reactivity: Human, Mouse
Details: Rabbit IgG Polyclonal
Applications: WB, Flow, ICC/IF
Western Blot: PARP Antibody [NBP3-09070]
(4)
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Potent PARP-1 inhibitor

Chemical Name: 5'-Deoxy-5'-[4-[2-[(2,3-Dihydro-1-oxo-1H-isoindol-4-yl)amino]-2-oxoethyl]-1-piperazinyl]-5'-oxoadenosine dihydrochloride
Purity: ≥98%
Potent PARP-1 inhibitor
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Potent fluorescent PARP inhibitor; cell permeable

Alternate Names: AZD2281-BDY FL,Olaparib-BDY FL
Chemical Name: (T-4)-[4-[[3-[[4-[3-[5-[(3,5-Dimethyl-2H-pyrrol-2-ylidene-κN)methyl]-1H-pyrrol-2-yl-κN-1-oxopropyl]-1-piperazinyl]carbonyl]-4-fluorophenyl]methyl]-1(2H)-phthalazinonato]difluoroboron
Purity: ≥90%
Potent fluorescent PARP inhibitor; cell permeable
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Potent PARP inhibitor

Chemical Name: 4-[[3-[[4-(Cyclopropylcarbonyl)-1-piperazinyl]carbonyl]-4-fluorophenyl]methyl]-1(2H)-phthalazinone
Purity: ≥98%
Potent PARP inhibitor
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Potent PARP inhibitor

Chemical Name: N-(5,6-Dihydro-6-oxo-2-phenanthridinyl)-2-acetamide hydrochloride
Purity: ≥98%
Potent PARP inhibitor
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Potent PARP inhibitor; orally bioavailable

Chemical Name: 4-[[4-Fluoro-3-[(4-methoxy-1-piperidinyl)carbonyl]phenyl]methyl]-1(2H)-phthalazinone
Purity: ≥98%
Potent PARP inhibitor; orally bioavailable
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PARP inhibitor

Alternate Names: CO-338
Chemical Name: 8-Fluoro-1,3,4,5-tetrahydro-2-[4-[(methylamino)methyl]phenyl]-6H-pyrrolo[4,3,2,ef][2]benzazepin-6-one (1S,4R)-7,7-dimethyl-2-oxobicyclo[2.2.1]heptane-1-methanesulfonic acid
Purity: ≥98%
PARP inhibitor
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Selective PARP-10 inhibitor

Chemical Name: 4,4'-Oxybis[benzamide]
Purity: ≥98%
Selective PARP-10 inhibitor
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PARP inhibitor; cytoprotectant

Chemical Name: N-[2-Hydroxy-3-(1-piperidinyl)propoxy]-3-pyridinecarboximidamide dihydrochloride
Purity: ≥98%
PARP inhibitor; cytoprotectant
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Selective allosteric PARP14 inhibitor

Chemical Name: N-[2-(9H-Carbazol-1-yl)phenyl]acetamide
Purity: ≥98%
Selective allosteric PARP14 inhibitor
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