29 results for "Dopamine D3 R/DRD3" in Products

Dopamine D3 R/DRD3 Products

DRD3 is the D3 subtype of the five (D1-D5) dopamine receptors. The activity of the D3 subtype receptor is mediated by G proteins which inhibit adenylyl cyclase. It is localized to the limbic areas of the brain, which are associated with cognitive, emotional, and endocrine functions. Genetic variations may be associated with susceptibility to hereditary essential tremor 1. Alternative splicing results in transcript variants encoding different isoforms. This variant represents the predominant transcript and encodes the longer isoform (a).

Dopamine precursor

Alternate Names: Levodopa
Chemical Name: L-3,4-Dihydroxyphenylalanine
Purity: ≥98%
Dopamine precursor
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High affinity D3 agonist (D3 ≥ D2 > D4)

Chemical Name: (4aR,10bR)-3,4a,4,10b-Tetrahydro-4-propyl-2H,5H-[1]benzopyrano-[4,3-b]-1,4-oxazin-9-ol hydrochloride
Purity: ≥98%
High affinity D3 agonist (D3 ≥ D2 > D4)
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Potent and selective D2 and D3 antagonist

Chemical Name: 3,5-Dichloro-N-[[(2S)-1-ethyl-2-pyrrolidinyl]methyl]-2-hydroxy-6-methoxybenzamide
Purity: ≥98%
Potent and selective D2 and D3 antagonist
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D2 and D3 antagonist (D3 > D2)

Alternate Names: (-)-Eticlopride
Chemical Name: 3-Chloro-5-ethyl-N-[[(2S)-1-ethyl-2-pyrrolidinyl)methyl]-6-hydroxy-2-methoxy-benzamide hydrochloride
Purity: ≥98%
D2 and D3 antagonist (D3 > D2)
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D2-like agonist (D2>D3>D4)

Chemical Name: (5'a)-2-Bromo-12'-hydroxy-2'-(1-methylethyl)-5'-(2-methylpropyl)ergotaman-3',6',18-trione mesylate
Purity: ≥98%
D2-like agonist (D2>D3>D4)
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Selective D3 agonist

Chemical Name: (S)-2-Amino-4,5,6,7-tetrahydro-6-(propylamino)benzothiazole dihydrochloride
Purity: ≥99%
Selective D3 agonist
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Caged dopamine; photolysed by UV light

Purity: ≥98%
Caged dopamine; photolysed by UV light
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Reactivity: Human, Mouse, Rat
Details: Rabbit Polyclonal
Applications: WB, ELISA, ICC/IF, IP, DB
Western Blot: Dopamine D3R/DRD3 Antibody [NBP3-12391]
(2)
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Potent 5-HT2 antagonist; also 5-HT3, H1 and α2 antagonist; antidepressant

Alternate Names: Org 3770,6-Azamianserin
Chemical Name: 1,2,3,4,10,14b-Hexahydro-2-methylpyrazino[2,1-a]pyrido[2,3-c][2]benzazepine
Purity: ≥98%
Potent 5-HT2 antagonist; also 5-HT3, H1 and α2 antagonist; antidepressant
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Potent and selective D3 antagonist

Chemical Name: N-[4-[4-(2,3-Dichlorophenyl)-1-piperazinyl]butyl]-9H-fluorene-2-carboxamide
Purity: ≥98%
Potent and selective D3 antagonist
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Non-selective 5-HT, dopamine, adrenalin and histamine receptor antagonist; antipsychotic agent

Chemical Name: (3aR*,12bR*)-5-Chloro-2,3,3a,12b-tetrahydro-2-methyl-1H-dibenz[2,3:6,7]oxepino[4,5-c]pyrrole maleate
Purity: ≥98%
Non-selective 5-HT, dopamine, adrenalin and histamine receptor antagonist; antipsychotic agent
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Selective D3 antagonist

Chemical Name: N-[(2E)-4-[4-(2,3-Dichlorophenyl)-1-piperazinyl]-2-buten-1-yl]-4-(2-pyridyl)-benzamide dihydrochloride
Purity: ≥98%
Selective D3 antagonist
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D2 and D3 agonist

Alternate Names: N 0923
Chemical Name: (6S)-5,6,7,8-Tetrahydro-6-[propyl[2-(2-thienyl)ethyl]amino]-1-naphthalenol hydrochloride
Purity: ≥99%
D2 and D3 agonist
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Selective D3 antagonist

Chemical Name: N-[trans-4-[2-(6-Cyano-3,4-dihydro-2(1H)-isoquinolinyl)ethyl]cyclohexyl]-4-quinolinecarboxamide dihydrochloride
Purity: ≥98%
Selective D3 antagonist
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Recombinant Monoclonal Antibody

Reactivity: Human, Mouse, Rat
Details: Rabbit IgG Monoclonal Clone #5L1P4
Applications: WB
Western Blot: Dopamine D3R/DRD3 Antibody (5L1P4) [NBP3-16443]
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Recombinant Monoclonal Antibody

Reactivity: Human, Mouse, Rat
Details: Rabbit IgG Monoclonal Clone #JE33-33
Applications: WB
Dopamine D3R/DRD3 Antibody (JE33-33)
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Recombinant Monoclonal Antibody

Reactivity: Human, Mouse, Rat
Details: Rabbit IgG Monoclonal Clone #SR1747
Applications: WB
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Reactivity: Human
Sensitivity: 0.19 ng/mL
Assay Range: 0.31 - 20 ng/mL
Applications: ELISA
Human Dopamine D3R/DRD3 ELISA Kit (Colorimetric)
(2)
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Reactivity: Rat
Sensitivity: 37.50 pg/mL
Assay Range: 62.50-4000 pg/mL
Applications: ELISA
Rat Dopamine D3R/DRD3 ELISA Kit (Chemiluminescence)
(2)
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Reactivity: Mouse
Sensitivity: 0.10 ng/mL
Assay Range: 0.16 - 10 ng/mL
Applications: ELISA
Mouse Dopamine D3R/DRD3 ELISA Kit (Colorimetric)
(2)
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Reactivity: Rat
Sensitivity: 0.19 ng/mL
Assay Range: 0.31 - 20 ng/mL
Applications: ELISA
Rat Dopamine D3R/DRD3 ELISA Kit (Colorimetric)
(2)
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Reactivity: Mouse, Rat
Details: Rabbit IgG Polyclonal
Applications: WB
Dopamine D3R/DRD3 Antibody - Azide and BSA Free
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