20 results for "alpha-1B Adrenergic R/ADRA1B Small Molecules and Peptides" in Products
alpha-1B Adrenergic R/ADRA1B Small Molecules and Peptides
ADRA1B, also known as the alpha-1B-adrenergic receptor, is a 7TM catecholamine receptor with selectivity for epinephrine and norepinephrine. ADRA1B functions in diverse settings including vasoconstriction and myocardial contractility, neuronal dopaminergic responses, dendritic cell migration and inflammatory responses, and neuroendocrine regulation...
α1 and α2B antagonist; also MT3 antagonist
| Chemical Name: | 1-(4-Amino-6,7-dimethoxy-2-quinazolinyl)-4-(2-furanylcarbonyl)piperazine hydrochloride |
| Purity: | ≥98% |
α1 agonist
| Chemical Name: | (R)-(-)-1-(3-Hydroxyphenyl)-2-methylaminoethanol hydrochloride |
| Purity: | ≥98% |
Potent and non-selective β antagonist; also potent α1 antagonist
| Alternate Names: | BM 14190 |
| Chemical Name: | 1-(9H-Carbazol-4-yloxy)-3-[[2-(2-methoxyphenoxy)ethyl]amino]-2-propanol |
| Purity: | ≥98% |
Selective α1 agonist
| Chemical Name: | 2-(2-Cyclopropylphenoxymethyl)imidazoline hydrochloride |
| Purity: | ≥98% |
α2 agonist. Also I1 ligand
| Chemical Name: | 2-[(2,6-Dichlorophenyl)amino-2-imidazoline hydrochloride |
| Purity: | ≥98% |
α1 antagonist; PGK1 activator
| Chemical Name: | 1-(4-Amino-6,7-dimethoxy-2-quinazolinyl)-4-[(tetrahydro-2-furanyl)carbonyl]-piperazine hydrochloride |
| Purity: | ≥98% |
Non-selective 5-HT, dopamine, adrenalin and histamine receptor antagonist; antipsychotic agent
| Chemical Name: | (3aR*,12bR*)-5-Chloro-2,3,3a,12b-tetrahydro-2-methyl-1H-dibenz[2,3:6,7]oxepino[4,5-c]pyrrole maleate |
| Purity: | ≥98% |
Potent and selective α2 antagonist
| Chemical Name: | 6-Chloro-N-methyl-2,3,4,5-tetrahydro-1-H-3-benzazepine hydrochloride |
| Purity: | ≥98% |
Highly selective α1 antagonist
| Alternate Names: | BE 2254 |
| Chemical Name: | 2-{[β-(4-Hydroxyphenyl)ethyl]aminomethyl}-1-tetralone hydrochloride |
| Purity: | ≥98% |
α1 antagonist
| Alternate Names: | UK 33274 |
| Chemical Name: | 4-Amino-2-[4-(1,4-benzodioxan-2-carbonyl)piperazin-1-yl]-6,7-dimethoxyquinazoline methanesulfonate |
| Purity: | ≥98% |
Selective α1A antagonist
| Chemical Name: | 5-[(2R)-2-[[2-(2-Ethoxyphenoxy)ethyl]amino]propyl]-2-methoxybenzenesulfonamide hydrochloride |
| Purity: | ≥98% |
Adrenergic α receptor antagonist; antihypertensive
| Chemical Name: | 3-[[(4,5-Dihydro-1H-imidazol-2-yl)methyl](4-methylphenyl)amino]phenol methanesulfonate |
| Purity: | ≥98% |
GluN2B-selective NMDA antagonist
| Chemical Name: | (αR,βS)-α-(4-Hydroxyphenyl)-β-methyl-4-(phenylmethyl)-1-piperidinepropanol maleate |
| Purity: | ≥98% |
Dopamine antagonist with some D4 selectivity; also 5-HT2A/2C antagonist
| Chemical Name: | 8-Chloro-11-(4-methyl-1-piperazinyl)-5H-dibenzo[b,e][1,4]diazepine |
| Purity: | ≥98% |
Dopamine antagonist; displays some D2 selectivity
| Chemical Name: | 4-[4-(4-Chlorophenyl)-4-hydroxy-1-piperidinyl]-1-(4-fluorophenyl)-1-butanone hydrochloride |
| Purity: | ≥98% |
5-HT4 agonist; stimulates intestinal ACh release
| Alternate Names: | R 51619 |
| Chemical Name: | (±)-4-Amino-5-chloro-N-[1-[(3R*,4S*)-3-(4-fluorophenoxy)propyl]-3-methoxy-4-piperidinyl]-2-methoxybenzamide |
| Purity: | ≥99% |
5-HT2A antagonist; also D2 antagonist; atypical antipsychotic
| Chemical Name: | 2-Methyl-4-(4-methyl-1-piperazinyl)-10H-thieno[2,3-b][1,5]benzodiazepine |
| Purity: | ≥98% |
5-HT2 antagonist; also D2 antagonist; atypical antipsychotic
| Alternate Names: | ICI 204,636 |
| Chemical Name: | 2-[2-(4-Dibenzo[b,f][1,4]thiazepin-11-yl-1-piperazinyl)ethoxy]ethanol hemifumarate |
| Purity: | ≥98% |
High affinity D2 and 5-HT1A receptor partial agonist; also 5-HT2A antagonist
| Chemical Name: | 7-[4-[4-(2,3-Dichlorophenyl)-1-piperazinyl]butoxy]-3,4-dihydro-2(1H)-quinolinone |
| Purity: | ≥99% |
Selective 5-HT1A agonist
| Alternate Names: | TVX Q 7821 |
| Chemical Name: | 2-[4-[4-(2-Pyrimidinyl)-1-piperazinyl]butyl]-1,2-benzisothiazol-3(2H)-one-1,1-dioxide |
| Purity: | ≥99% |
