Peptide Receptors

Peptide receptors constitute a large group of GPCRs that are activated by extracellular protein or peptide ligands. Endogenous peptide receptor ligands bind to the N' terminus and/or the 3 extracellular loops of the receptor. Consistent with the array of physiological roles of peptide receptors, the range of conditions in which they are dysregulated is vast and includes cardiovascular, endocrine and metabolic disorders.

Products for Peptide Receptors

Angiotensin Receptors Angiotensin Receptor Products	Motilin Receptor Motilin Receptor Products
Apelin Receptors (APJ) Apelin Receptor Agonists Apelin Receptor Antagonists	Neuromedin U Receptors (NMU₁, NMU₂) Neuromedin U Receptor Products
Bombesin Receptors (Bombesin Receptors) Bombesin Receptor Agonists Bombesin Receptor Antagonists	Neuropeptide FF/AF Receptors Neuropeptide FF/AF Receptor Agonists Neuropeptide FF/AF Receptor Antagonists
Bradykinin Receptors (BDKRB1, BDKRB2) Bradykinin Receptor Agonists Bradykinin Receptor Antagonists	Neuropeptide S Receptors (NPSR1) Neuropeptide S Receptors Agonists Neuropeptide S Receptors Antagonists
Calcitonin and Related Receptors (Calcitonin and Related Receptors) Calcitonin and Related Receptor Agonists Calcitonin and Related Receptor Antagonists	Neurotensin Receptors (NTS₁, NTS₂, Sortilin) Neurotensin Receptor Agonists Neurotensin Receptor Partial Agonists Neurotensin Receptor Antagonists
Cholecystokinin Receptors Cholecystokinin Receptor Products	NPY Receptors (NPY1R, NPY2R, NPY4R, NPY5R) NPY Receptor Agonists NPY Receptor Antagonists
CRF Receptors CRF Receptor Products	Orexin Receptors Orexin Receptor Products
Endothelin Receptors Endothelin Receptor Products	Other Peptide Receptors Other Peptide Receptor Products
Formyl Peptide Receptors (FPR1, FPR2, FPR3) Formyl Peptide Receptor Agonists Formyl Peptide Receptor Antagonists	Oxytocin Receptors (OXTR) Oxytocin Receptor Agonists Oxytocin Receptor Antagonists
Galanin Receptors (GAL₁, GAL₂, GAL₃) Galanin Receptor Agonists Galanin Receptor Antagonists	PACAP Receptors PACAP Receptor Agonists PACAP Receptor Antagonists
Ghrelin Receptors (GHSR) Ghrelin Receptor Agonists Ghrelin Receptor Inverse Agonists Ghrelin Receptor Antagonists Other Ghrelin Receptor Peptides	Parathyroid Hormone Receptors (PTH1R, PTH2R) Parathyroid Hormone Receptor Agonists
Glucagon and Related Receptors Glucagon and Related Receptor Products	Protease-Activated Receptors (PARs) Protease-Activated Receptor Agonists Protease-Activated Receptor Antagonists Protease-Activated Receptor Inhibitors
Gonadotropin-Releasing Hormone Receptors (GnRHR) Gonadotropin-Releasing Hormone Receptor Antagonist	Somatostatin (sst) Receptors (SSTRs) Somatostatin (sst) Receptor Agonists Somatostatin (sst) Receptor Antagonists Additional Somatostatin Receptor Peptides
GPR171 (GPR171) GPR171 Agonists GPR171 Antagonists	Tachykinin Receptors Tachykinin Receptor Products
GPR83 (GPR83) GPR83 Agonists	Thyrotropin-Releasing Hormone Receptors TRHR Products
Kisspeptin Receptor (KISS1R) Kisspeptin Receptor Agonists Kisspeptin Receptor Antagonists	Urotensin-II Receptors (Urotensin-II R) Urotensin-II Receptor Antagonists
Mas-Related G Protein-Coupled Receptors (MRGPRs) Mas-Related G Protein-Coupled Receptors Agonists Mas-Related G Protein-Coupled Receptors Antagonists Mas-Related G Protein-Coupled Receptors Modulators	Vasopressin Receptors (V_1A, V_1B, V₂) Vasopressin Receptor Agonists Vasopressin Receptor Antagonists
Melanin-concentrating Hormone Receptors (MCHR1, MCHR2) Melanin-concentrating Hormone Receptor Agonists Melanin-concentrating Hormone Receptor Antagonists	VIP Receptors (VPAC₁, VPAC₂) VIP Receptor Agonists VIP Receptor Antagonists
Melanocortin (MC) Receptors Melanocortin (MC) Receptor Agonists Melanocortin (MC) Receptor Antagonists Additional Melanocortin (MC) Receptor Peptides